Patent · US Expired

9-OXO-15 .xi.-HYDROXY-20-ALKYLIDENEPROST-13(TRANS)-ENOIC ACID DERIVATIVES

US4064351A · kind A · utility

31Cited by
1References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 22, 1976
Grant dateDec 20, 1977
Priority date
Expiry dateDec 22, 1996

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/4015
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Prostanoic acid derivatives having the formula ##STR1## wherein A represents ethylene group or cis-vinylene group, R.sup.1 and R.sup.2 may be the same or different and each represents hydrogen atom or an alkyl group having 1-3 carbon atoms, R.sup.3 and R.sup.4 may be the same or different and each represents an alkyl group having 1-3 carbon atoms and R.sup.5 represents hydrogen atom or hydroxyl group and the pharmaceutically acceptable salts thereof and a process for the preparation thereof. The compounds are useful as anti-ulcerogenic or bronchodilating agents and may be prepared by oxidizing 9.xi.-hydroxy-15.xi.-protected-hydroxy-20-alkylideneprost-13(trans)-enoic acid derivatives.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.