Styrylsulfonylamidines
US4096183A · kind A · utility
1Cited by
0References
39Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Aug 19, 1977 |
| Grant date | Jun 20, 1978 |
| Priority date | — |
| Expiry date | Aug 19, 1997 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P25/04
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Styrylamidines are prepared by treating styrylsulfonylamidines with base. The styrylamidines are effective in the prevention of aggregation of blood platelets and as analgesics. Compounds of the invention are also useful as anticonvulsants, diuretics and antihypertensive agents. The styrylsulfonylamidines of the invention which serve as precursors to the styrylamidines also have analgesic properties. Illustrative of the styrylamidines of the present invention are 4-amino-N-(4-aminostyryl)benzamidine and N-(3,4-dichlorostyryl)acetamidine. An example of a styrylsulfonylamidine is N-(styrylsulfonyl)acetamidine.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.