Patent · US Expired

Method for inhibiting emesis and compositions therefor

US4101662A · kind A · utility

7Cited by
3References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 3, 1973
Grant dateJul 18, 1978
Priority date
Expiry dateMay 3, 1993

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D211/32
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

1,4-(3-)Disubstituted piperidines are disclosed which have useful antiemetic properties. The compounds have the general formula: ##STR1## wherein R is halogen, R.sup.1 is hydrogen and halogen, n is a positive integer from 2-4 and A is --C(O)-- and --CHOH--. The pharmaceutically acceptable acid addition salts of the basic compounds are particularly useful as antiemetics.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.