Triazolyl benzophenones
US4111950A · kind A · utility
Assignee
Inventors
Key dates
| Filing date | Feb 4, 1977 |
| Grant date | Sep 5, 1978 |
| Priority date | — |
| Expiry date | Feb 4, 1997 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC09B29/32
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Compounds of the class of 6-phenyl-4H-s-triazolo[1,5-a][1,4]benzodiazepine-2-carboxamides, their 5-oxides and their pharmaceutically acceptable acid addition salts have valuable pharmacological properties and are active ingredients for therapeutic compositions. In particular, these new compounds have an anti-convulsive and anti-aggressive action and inhibit somatic reflexes. Specific embodiments are N,N-dimethyl-6-phenyl-8-chloro-4H-s-triazolo[1,5-a][1,4]benzodiazepine-2-c arboxamide, 6-(o-fluorophenyl)-8-chloro-4H-s-triazolo[1,5-a][1,4]benzodiazepine-2-carb oxamide, N,N-dimethyl-6-(o-fluorophenyl)-8-chloro-4H-s-triazolo[1,5-a][1,4]benzodia zepine-2-carboxamide and N,N-dimethyl-6-(o-chlorophenyl)-8-chloro-4H-s-triazolo[1,5-a][1,4]benzodia zepine-2-carboxamide.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.