Carbohydrate derivatives of milbemycin and processes therefor
US4134973A · kind A · utility
31Cited by
3References
6Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Apr 11, 1977 |
| Grant date | Jan 16, 1979 |
| Priority date | — |
| Expiry date | Apr 11, 1997 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07H17/08
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Carbohydrate derivatives of the antibiotic substance milbemycin, also identified as B-41, and of 13-hydroxy milbemycin are prepared. The carbohydrate groups are attached to the available hydroxy groups of milbemycin and to the hydroxy group synthesized at the 13-position. The reactions may be made selectively such that more than one carbohydrate group may be attached to a single position, or that multiple carbohydrate groups may be attached at different positions on the molecule. The described carbohydrate derivatives have antiparasitic activity.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.