Patent · US Expired

Novel imidazobenzoxazines

US4145419A · kind A · utility

10Cited by
1References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 1, 1977
Grant dateMar 20, 1979
Priority date
Expiry dateAug 1, 1997

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D265/36
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel imidazobenzoxazines of the formula ##STR1## wherein X is selected from the group consisting of hydrogen, nitro, NH.sub.2 and a protected amino Z is selected from the group consisting of --COOR, and ##STR2## R is selected from the group consisting of hydrogen, alkyl of 1 to 5 carbon atoms, ##STR3## alkali metal, alkaline earth metal, magnesium, aluminum and nitrogen bases, n is 1,2 or 3, R.sub.1 and R.sub.2 individually are selected from the group consisting of hydrogen and alkyl of 1 to 5 carbon atoms and taken together with the nitrogen atom to which they are attached form a saturated heterocyclic ring of 4 to 6 carbon atoms optionally interrupted by another heteroatom which may optionally be substituted with alkyl of 1 to 5 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts having antiallergic and bronchodilatory activity and their preparation.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.