Azetidine compounds and process for production
US4163855A · kind A · utility
3Cited by
0References
4Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Mar 23, 1978 |
| Grant date | Aug 7, 1979 |
| Priority date | — |
| Expiry date | Mar 23, 1998 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D213/55
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
Novel azetidine, and particularly 2-pyridyl-azetidine, compounds are disclosed. These compounds are produced from amino-esters by a sequence comprising conversion to the sulfonamide, reduction of the ester to the alcohol, sulfonation of the resultant alcohol and cylization to the N-sulfonylazetidine. This azetidine compound may then be transformed, as desired, to various N-derivatives by substitution of hydrogen or other univalent organic groups on the secondary amine of the azetidine ring.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.