Patent · US Expired

Oxazolinoazetidinylbutyric acid derivatives

US4183855A · kind A · utility

11Cited by
0References
1Claims
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Assignee

Inventors

Key dates

Filing dateFeb 24, 1978
Grant dateJan 15, 1980
Priority date
Expiry dateFeb 24, 1998

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D505/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Intermediates (I) for preparing a potent antibacterial, 1-oxadethiacephalosporin, are shown by the following formula ##STR1## (wherein R is a group of acyl-minus-carbonyl derived from a carboxylic or carbonic acid; PA1 COB is carboxy or protected carboxy; PA1 X is hydrogen or a nucleophilic group; PA1 Y is a nucleophilic group; and PA1 Z is a leaving group) and prepared from the corresponding exomethylene compound (II) by addition of a compound of formula: Y-Z (in which Y and Z are as defined above).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.