Patent · US Expired

Hexahydroazepine, piperidine and pyrrolidine derivatives

US4197239A · kind A · utility

2Cited by
0References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 15, 1978
Grant dateApr 8, 1980
Priority date
Expiry dateNov 15, 1998

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D223/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention concerns novel 2-oxo-hexahydroazepine, -piperidine and -pyrrolidine of formula I ##STR1## where n is 2,3 or 4, R is hydrogen, lower alkyl or aryl(lower)alkyl and R.sup.1 is lower alkyl. The compounds may be aromatized and the aromatized compounds converted to 3,3-disubstituted-hexahydroazepine, -piperidine and -pyrrolidine compounds having pharmacological activity, particularly analgesic activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.