Patent · US Expired

Alkyl derivatives of C-076 compounds

US4200581A · kind A · utility

38Cited by
1References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 4, 1978
Grant dateApr 29, 1980
Priority date
Expiry dateAug 4, 1998

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P33/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Derivatives of C-076, a series of macrolides are described, in which the substituents are hydrocarbon groups. The hydrocarbon groups generally are alkyl groups which may be straight or branched and may optionally be substituted with phenyl. The substituted C-076 compounds are prepared by various procedures depending upon the position of the reaction site, and the particular C-076 compound being substituted. The compounds have profound anthelmintic, insecticidal, ectoparasiticidal and acaracidal activity and compositions for such uses are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.