Azepino [1,2,3-lm]-.beta.-carboline compounds and pharmaceutical composition thereof
US4228168A · kind A · utility
4Cited by
0References
7Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Nov 2, 1979 |
| Grant date | Oct 14, 1980 |
| Priority date | — |
| Expiry date | Nov 2, 1999 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D209/16
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
An azepino[1,2,3-lm]-.beta.-carboline compound of the formula: ##STR1## wherein R.sup.1 is hydrogen, cycloalkyl of 3 to 7 carbon atoms, phenyl, hydroxy, alkoxycarbonyl of 2 or 3 carbon atoms or alkanoyl of 2 or 3 carbon atoms, and A is single bond or straight or branched alkylene of one to 5 carbon atoms. Several methods of preparing the compound [I] are disclosed. The compound [I] and a pharmaceutical acceptable acid addition salt thereof have a potent anti-anoxic activity.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.