Patent · US Expired

Drug excipient of silicone rubber

US4230686A · kind A · utility

21Cited by
6References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 23, 1976
Grant dateOct 28, 1980
Priority date
Expiry dateDec 23, 1996

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC08G77/20
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Nontoxic sustained release pharmaceutical compositions containing one or more nonionic, lipophilic drugs in a cured low temperature vulcanizable (LTV) silicone elastomer excipient are prepared substantially free of toxic vulcanizing agents or drug-reactive by-products in the elastomeric material by curing an admixture of the drug or drug containing core, LTV-methylvinylsiloxane units containing linear dimethylpolysiloxane and a dimethylpolysiloxane crosslinking composition containing silicon linked H atoms using a noble metal-based catalyst. The resultant compositions are characterized by good physical properties and a constant rate of drug release in the body over long periods of time.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.