Patent · US Expired

2 -Alkylsulphonyl-7,8-dihydro-5-hydroxy-7-oxo-pyrido[2,3-d]pyrimidine-6-car boxylic acid derivatives

US4236004A · kind A · utility

3Cited by
2References
2Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 29, 1979
Grant dateNov 25, 1980
Priority date
Expiry dateOct 29, 1999

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D498/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

2-Alkylsulfonyl-7,8-dihydro-5-hydroxy-7-oxo-pyrido[2,3-d]pyrimidine-6-carbo xylic acid derivatives are intermediates useful in the production of 7,8-dihydro-2-amino or alkoxy-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives which are gastric anti-secretory agents for treatment of peptic ulcer disease and generally anti-allergic agents useful in the treatment of atopic immediate hypersensitivity reactions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.