Patent · US Expired

Prostaglandin analogues

US4241074A · kind A · utility

1Cited by
1References
40Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 14, 1979
Grant dateDec 23, 1980
Priority date
Expiry dateJun 14, 1999

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D233/76
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A compound of the formula (I): ##STR1## wherein: X is O, S or H; PA1 Y is --CH.sub.2 --CH--, --CH.dbd.CH-- or --C.dbd.C--; PA1 n is 1 to 7; PA1 R.sub.1 is C.sub.1-4 alkyl; PA1 R.sub.3 is hydroxy or protected hydroxy; PA1 R.sub.4 is C.sub.1-9 alkyl, C.sub.3-8 cycloalkyl or C.sub.3-8 cycloalkyl--C.sub.1-6 alkyl; or PA1 R.sub.2 and R.sub.4 taken with the carbon atom to which they are joined represent a C.sub.5-8 cycloalkyl group; and PA1 R.sub.5 is hydrogen or C.sub.1-6 alkyl; and salts thereof has useful pharmaceutical activity including bronchodilator activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.