Patent · US Expired

Substituted benzonitriles having antiviral activity

US4254144A · kind A · utility

2Cited by
10References
49Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJan 25, 1980
Grant dateMar 3, 1981
Priority date
Expiry dateJan 25, 2000

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C317/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Substituted benzonitriles are disclosed having the formula ##STR1## wherein X represents O or S; R.sub.1 represents bromo, chloro, fluoro, phenoxy, loweralkylthio, loweralkylsulfinyl, loweralkylsulfonyl, loweralkylaminosulfonyl, diloweralkylaminosulfonyl or benzoyl; and R.sub.2 represents hydrogen, bromo, chloro or fluoro with the proviso that R.sub.2 is hydrogen when R.sub.1 is a substituent other than bromo, chloro or fluoro. The compounds of the invention exhibit antiviral activity. Methods of use based on the antiviral activity of the compounds are also disclosed, as well as compositions which comprise a carrier in combination with a suitable antiviral active compound.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.