Patent · US Expired

Acetoxymethyl penam compounds as .beta.-lactamase inhibitors

US4256733A · kind A · utility

8Cited by
0References
22Claims
0Family size

Assignee

Inventor

Key dates

Filing dateSep 26, 1979
Grant dateMar 17, 1981
Priority date
Expiry dateSep 26, 1999

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

2.beta.-Acetoxymethyl-2.alpha.-methyl-(5R)penam-3.alpha.-carboxylic acid 1,1-dioxide, pharmaceutically-acceptable salts thereof and esters thereof readily hydrolyzable in vivo; pharmaceutical compositions containing 2.beta.-acetoxymethyl-2.alpha.-methyl-(5R)penam-3.alpha.-carboxylic acid 1,1-dioxide or salt or ester thereof; and method of enhancing the effectiveness of a .beta.-lactam antibiotic using 2.beta.-acetoxymethyl-2.alpha.-methyl-(5R)penam-3.alpha.-carboxylic acid 1,1-dioxide or salt or ester thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.