Patent · US Expired

Pyrido[1,2-A]pyrimidine derivatives and method of analgesic treatment

US4291036A · kind A · utility

7Cited by
4References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 14, 1980
Grant dateSep 22, 1981
Priority date
Expiry dateMar 14, 2000

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P29/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of the formula ##STR1## or pharmaceutically acceptable acid-addition or quaternart ammonium salts thereof PA0 wherein PA0 R is hydroxy, carboxy, lower alkoxycarbonyl, benzyloxycarbonyl, phenoxycarbonyl, carbamoyl, N-loweralkyl-carbamoyl, N,N-dilower-alkyl-carbamoyl, carboazido, carbohydrazido or cyano; PA0 R.sup.2 is C.sub.1 to C.sub.6 alkyl; PA0 R.sup.3 is C.sub.1 to C.sub.6 alkyl or benzyl; and PA0 R.sup.4 is a single electron pair, hydrogen or lower alkyl; and the dotted lines represent saturated or unsaturated bonds, are disclosed with analgesic properties.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.