Patent · US Expired

Derivatives of A-30912A nucleus

US4293489A · kind A · utility

44Cited by
6References
40Claims
0Family size

Assignee

Inventor

Key dates

Filing dateAug 25, 1980
Grant dateOct 6, 1981
Priority date
Expiry dateAug 25, 2000

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12R2001/62
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of the formula ##STR1## wherein R.sup.1 is a group of the formula: ##STR2## wherein A is divalent oxygen, sulfur, sulfinyl, or sulfonyl; A.sup.1 is divalent oxygen, sulfur, sulfinyl, sulfonyl or --NH--; X is hydrogen, chloro, bromo, iodo, nitro, C.sub.1 --C.sub.3 alkyl, hydroxy, C.sub.1 -C.sub.3 alkoxy, mercapto, C.sub.1 -C.sub.3 alkylthio, carbamyl or C.sub.1 -C.sub.3 alkylcarbamyl; X.sup.1 is chloro, bromo or iodo; R.sup.2 is hydrogen, C.sub.1 -C.sub.18 alkyl or C.sub.2 -C.sub.18 alkenyl; W is C.sub.1 -C.sub.10 alkylene or C.sub.2 -C.sub.10 alkenylene; m, n and p are 0 or 1, but if m=0, n must=0; provided: that the sum of the carbon atoms in the R.sup.2 and W groups must be greater than 4 but cannot exceed 21; that when X is mercapto. A and A.sup.1 cannot be sulfinyl or sulfonyl; and that when A and A.sup.1 are sulfinyl or sulfonyl, they must be in equal oxidation states.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.