8-(5-Pyrimidinecarboxamide)nor-tropane derivatives
US4321378A · kind A · utility
29Cited by
2References
6Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Apr 16, 1981 |
| Grant date | Mar 23, 1982 |
| Priority date | — |
| Expiry date | Apr 16, 2001 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D451/04
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.