Patent · US Expired

Anthracycline glycosides, their preparation, use and compositions thereof

US4322412A · kind A · utility

1Cited by
3References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 14, 1980
Grant dateMar 30, 1982
Priority date
Expiry dateJul 14, 2000

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

There are disclosed compounds which exhibit anti-tumor activity. These compounds are of the formula I: ##STR1## wherein R.sub.1 is hydrogen, hydroxy or methoxy, R.sub.2 is hydrogen or hydroxy, and each of R.sub.3 and R.sub.4 independently is hydrogen or methyl, with the proviso that R.sub.3 and R.sub.4 are not simultaneously hydrogen, and pharmaceutically acceptable acid addition salts thereof. Also disclosed are processes for producing and using said compounds and therapeutic compositions containing same.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.