Patent · US Expired

Pyrrolo(2,3-d)carbazole derivatives, compositions and use

US4362739A · kind A · utility

9Cited by
1References
19Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMay 4, 1981
Grant dateDec 7, 1982
Priority date
Expiry dateMay 4, 2001

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention relates to alkyl pyrrolo(2,3-d) carbazole-6-carboxylates having antianoxic, psychotropic and hemodynamic properties and to addition salts thereof; and to preparation of the same by a synthesis sequence starting from a tryptamine and a 3-halopyruvate and involving a rearrangement of an addition compound with an aldehyde, said rearrangement being effected by Nb-alkylation of the aforementioned addition compound; and to pharmaceutical compositions containing the same; and to tetrahydroazepinoindoles used in the preparation of the same.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.