Bis-esters of alkanediols as antibacterial agents
US4364957A · kind A · utility
2Cited by
3References
9Claims
0Family size
Assignee
Inventor
Key dates
| Filing date | Feb 20, 1981 |
| Grant date | Dec 21, 1982 |
| Priority date | — |
| Expiry date | Feb 20, 2001 |
Classification
- Technology area (CPC A)Human Necessities
- CPC primaryA61P31/04
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
6-Acylaminopenicillanoyloxymethyl esters and 1-(6-acylaminopenicillanoyloxy)ethyl esters of 2-beta-acetoxymethyl-2-alpha-methyl-(5R)penam-3-alpha-carboxylic acid 1,1-dioxide are useful as antibacterial agents. The 6-aminopenicillanoyloxymethyl ester, the 1-(6-aminopenicillanoyloxy)ethyl ester and certain other mono-substituted methyl and ethyl esters of 2-beta-acetoxymethyl-2-alpha-methyl-(5R)penam-3-alpha-carboxylic acid 1,1-dioxide are useful intermediates to the aforesaid antibacterial agents.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.