Patent · US Expired

Cephalosporin analogs for oral use

US4376770A · kind A · utility

1Cited by
0References
20Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 23, 1981
Grant dateMar 15, 1983
Priority date
Expiry dateJul 23, 2001

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P31/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

7.beta.-(2-Cyano-aliphatic acylamino)-7.alpha.-methoxy-3-heterocyclic thiomethyl-1-dethia-1-oxa-3-cephem-4-carboxylic acids and salts or pharmacologically acceptable esters generically represented by the following formula are potent antibacterials and esters are prospective oral drugs: ##STR1## (wherein A is a lower alkyl, lower alkenyl or lower alkynyl group; PA1 B is a hydrogen atom, salt forming atom, salt forming group or physiologically hydrolyzable ester group; and PA1 Het is a heterocyclic group).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.