Patent · US Expired

Novel oximes

US4420478A · kind A · utility

4Cited by
2References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 9, 1979
Grant dateDec 13, 1983
Priority date
Expiry dateApr 9, 1999

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D277/587
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel syn isomers of oximes of 3-azidomethyl-7-amino-thiazolyl-cephalosporanic acids of the formula ##STR1## wherein R is selected from the group consisting of hydrogen, alkyl of 1 to 4 carbon atoms, unsaturated alkyl of 2 to 4 carbon atoms, benzoyl and --(CH.sub.2).sub.n --R.sub.1, n is an integer from 1 to 4, R.sub.1 is selected from the group consisting of NH.sub.2 and --COOA' and A' and A are selected from the group consisting of hydrogen, alkali metal, alkaline earth metal, magnesium, --NH.sub.4, an easily cleavable ester group and a non-toxic, pharmaceutically acceptable organic amine and their non-toxic, pharmaceutically acceptable acid addition salts having antibiotic activity and a novel process and novel intermediates for their preparation.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.