Patent · US Expired

Processes for the interconversion of avermectin compounds

US4423209A · kind A · utility

50Cited by
8References
4Claims
0Family size

Assignee

Inventor

Key dates

Filing dateFeb 26, 1982
Grant dateDec 27, 1983
Priority date
Expiry dateFeb 26, 2002

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07H19/01
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

There is disclosed a process for converting avermectin compounds (formerly identified as C-076 compounds) of the A-type, into avermectin compounds of the B-type. The process is carried out on the naturally occuring avermectin compounds as well as on derivatives thereof. The process involves selectively cleaving the 5-methoxy group, converting it into the hydroxy group, through the intermediate 5-keto group.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.