Azepino[4,5-d]indole derivatives and preparation thereof
US4428880A · kind A · utility
6Cited by
6References
7Claims
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Assignee
Inventor
Key dates
| Filing date | Sep 29, 1982 |
| Grant date | Jan 31, 1984 |
| Priority date | — |
| Expiry date | Sep 29, 2002 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D487/10
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
This invention relates to novel tetrahydroazepinoindoles used in the preparation of novel alkyl pyrrolo(2,3-d)carbazole-6-carboxylates and to addition salts thereof; and to preparation of the same by a synthesis sequence starting from a tryptamine and a 3-halopyruvate and involving a rearrangement of the reaction mixture, said rearrangement being effected by heating the reaction mixture in the presence of a base. The pyrrolo(2,3-d)carbazole final products have both antianoxic and psychotropic activities.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.