Patent · US Expired

Benzimidazole derivatives, process for the preparation thereof and pharmaceutical composition containing the same

US4430343A · kind A · utility

22Cited by
3References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 22, 1982
Grant dateFeb 7, 1984
Priority date
Expiry dateOct 22, 2002

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel benzimidazole derivatives of the formula: ##STR1## wherein R.sup.1 is an alkyl group having 1 to 3 carbon atoms, allyl group, propargyl group, or phenyl group; R.sup.2 is hydrogen atom or an alkyl group having 1 to 3 carbon atoms; and n is 2 or 3, or pharmaceutically acceptable acid addition salts thereof, which have excellent antihistaminic activities and are useful as antiallergics for various allergic diseases, and a process for the preparation thereof, and an antihistaminic composition containing the compound as an active ingredient.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.