Patent · US Expired

Naphthalenylthiazole derivatives

US4446150A · kind A · utility

1Cited by
3References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 21, 1982
Grant dateMay 1, 1984
Priority date
Expiry dateSep 21, 2002

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P3/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed herein are new aldose reductase inhibitors of the formula ##STR1## wherein R is ##STR2## wherein R.sup.1 is lower alkyl; R.sup.2 is halo and R.sup.3 is hydrogen, or R.sup.2 and R.sup.3 each is a substituent at positions 3, 4, 5 or 6 of the naphthalene ring selected from the group consisting of lower alkoxy, trihalomethyl, and halo; and R.sup.4 is lower alkyl. The derivatives are useful for treating or preventing diabetic complications.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.