Patent · US Expired

16.beta.-Methyl steroid process

US4451404A · kind A · utility

1Cited by
3References
26Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 9, 1983
Grant dateMay 29, 1984
Priority date
Expiry dateFeb 9, 2003

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07J17/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

.DELTA..sup.4 -3-keto, .DELTA..sup.1,4 -3-keto and 3.beta.-hydroxy 17-keto steroids (I) are transformed into the corresponding 16-.beta.-methyl-17-keto steroids (IV) by first activating the C-16 position, then methylating. By protecting the C-3 position of the .DELTA..sup.4 -3-keto and 3.beta.-hydroxy steroids the yields are greatly increased.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.