Patent · US Expired

Process for the preparation of 2-(thien-2-yl)- and 2-(thien-3-yl)-ethylamine derivatives

US4482718A · kind A · utility

3Cited by
3References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 29, 1982
Grant dateNov 13, 1984
Priority date
Expiry dateJun 29, 2002

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/65515
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides a process for the preparation of 2-(thien-2-yl)- and 2-(thien-3-yl)-ethylamine derivatives of the general formula: ##STR1## in which R.sub.1, in the 2-, 3-, 4- or 5-position, is a hydrogen or halogen atom, a nitro, carboxyl, cyano or amino group, a linear or branched alkyl or alkoxy radical or a heterocyclic or non-heterocyclic aromatic radical, which is optionally mono- or polysubstituted, the aminoethyl chain is in the 2- or 3-position, R.sub.2, R.sub.3 and R.sub.4, which are the same or different, are hydrogen atoms or heterocyclic or non-heterocyclic aromatic radicals, which are optionally mono- or polysubstituted, and Ar is a heterocyclic or non-heterocyclic aromatic radical, which is optionally mono- or polysubstituted.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.