Patent · US Expired

Isomerization of .beta.-lactam compounds

US4497742A · kind A · utility

1Cited by
2References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 24, 1982
Grant dateFeb 5, 1985
Priority date
Expiry dateFeb 24, 2002

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12R2001/465
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

Compounds of the formula (I): ##STR1## wherein R is an ethyl group which may optionally be substituted and n is 0 or 1, or a physiologically acceptable salt thereof, can be produced by subjecting to isomerization a compound of the formula (II): ##STR2## wherein R and n have the same meaning as defined above, or a salt thereof, by using a quaternary ammonium halide and are useful as a bactericide or disinfectant, and also a synergistic effect with penicillin and/or cephalosporin antibiotic agents. Among the compounds of the formula (I), compounds shown by the formula: ##STR3## wherein R.sub.6 is H or --SO.sub.3 H, as well as salts thereof, are novel.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.