Patent · US Expired

6H-indolo[2,1-c][1,4]benzodiazepines and 12-oxo derivatives useful as antihypertensives

US4529724A · kind A · utility

9Cited by
0References
10Claims
0Family size

Assignee

Inventor

Key dates

Filing dateOct 11, 1983
Grant dateJul 16, 1985
Priority date
Expiry dateOct 11, 2003

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the present invention are of the formula (I): ##STR1## wherein X is oxygen or two hydrogens, R.sup.1 is a variety of substituents or hydrogen and R.sup.2 is hydrogen, alkoxy, alkyl, CF.sub.3, halogen, NO.sub.2, OH or dialkylamino. The compounds are useful as blood pressure lowering agents and may be used in the treatment of hypertension. Also, part of the invention are pharmaceutical compositions and uses and intermediates for compounds of formula (I).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.