Patent · US Expired

Production of a cephalosporin by fermentation

US4533632A · kind A · utility

6Cited by
2References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 6, 1982
Grant dateAug 6, 1985
Priority date
Expiry dateAug 6, 2002

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC02F3/30
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

A process for greatly improving the yields of cephalosporin nucleus produced by fermentation is described. Cephalosporin C-producing microorganisms are fermented in the presence of an acetylesterase enzyme so that cephalosporin C formed is immediately converted into desacetyl cephalosporin C before any non-enzymic degradation occurs. Fermentation to produce desacetyl cephalosporin C enables yield increases of cephalosporin nucleus of about 40% to be realized, and greater increases are possible if the fermentation is extended. The preferred cephalosporin C-producing organism is Acremonium chrysogenum, and mutants thereof that are capable of producing esterases in situ. Alternatively, esterases obtained from a variety of other sources may be added or formed in situ, for example from a strain of Rhodosporidium.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.