Patent · US Expired

Analgesic dipeptide amides and method of use and composition thereof

US4533657A · kind A · utility

13Cited by
5References
14Claims
0Family size

Assignee

Inventor

Key dates

Filing dateSep 24, 1982
Grant dateAug 6, 1985
Priority date
Expiry dateSep 24, 2002

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K5/06078
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

A genus of dipeptide amides including as the preferred subgenus the dipeptide amides having the structural formula HTyrD-AlaNR.sub.2 R.sub.3 wherein R.sub.2 is phenylalkyl or substituted-phenylalkyl and R.sub.3 is hydrogen, alkyl, phenylalkyl, substituted-phenylalkyl or X-alkyl wherein X is an electronegative moiety are prepared by condensing the dipeptide with the amine or the amino acid with the amino acid amide and are useful as analgesics.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.