Patent · US Expired

4-Amino-5-bromo-2-methoxy-N-[8-(benzyl)]-8-azabicyclo[3.2.1] -3-YL-benzamide or a pharmacologically acceptable acid addition salt thereof

US4536580A · kind A · utility

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1References

1Claims

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Assignee

Delalande S.A. · FR

Inventors

Philippe L. Dostert · Chaville, FR
Thierry Imbert · Castres, FR
Bernard P. Bucher · Ville-d'Avray, FR

Key dates

Filing date	Jul 19, 1982
Grant date	Aug 20, 1985
Priority date	—
Expiry date	Jul 19, 2002

Classification

Technology area (CPC C)Chemistry; Metallurgy
CPC primaryC07D451/04
WIPO fieldOrganic fine chemistry
WIPO sectorChemistry

Abstract

There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.