Patent · US Expired

Amidine benzodiazepines, methods for their use and intermediates

US4547497A · kind A · utility

1Cited by
4References
20Claims
0Family size

Assignee

Inventor

Key dates

Filing dateApr 11, 1984
Grant dateOct 15, 1985
Priority date
Expiry dateApr 11, 2004

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Fused tetracyclic benzodiazepines of the formula (I): ##STR1## where R.sup.1 is an acyclic amine or cyclic amine such as 1-piperidine, 4-morpholine or 1-piperazine and R.sup.2 is H or a substituent as defined herein as useful as antiallergins. Also, methods for their synthesis, intermediate used in such synthesis, methods for use as medicaments and pharmaceutical compositions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.