Patent · US Expired

Pyrazolo[3,4-b]pyridine carboxylic acid esters and their pharmaceutical use

US4552883A · kind A · utility

8Cited by
3References
9Claims
0Family size

Assignee

Inventor

Key dates

Filing dateMay 19, 1983
Grant dateNov 12, 1985
Priority date
Expiry dateMay 19, 2003

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of the formula (I): ##STR1## wherein R.sup.1, R.sup.3, R.sup.4, R.sup.5 and R.sup.6 have defined values and the N-oxides at the 7-position of the pyrazolo[3,4-b]pyridine ring system and the pharmaceutically-acceptable acid-addition salts thereof, processes for their preparation and use, pharmaceutical compositions, and intermediates for preparing said compounds of the formula (I). The compounds of formula (I) are central nervous system depressants, for example anxiolytic agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.