Patent · US Expired

Isoxazolyl and isothiazolyl aromatase inhibitors

US4560695A · kind A · utility

1Cited by
5References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 18, 1984
Grant dateDec 24, 1985
Priority date
Expiry dateJun 18, 2004

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention provides certain isoxazole and isothiazole derivatives, their pharmaceutical formulations, and their use in inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.