Patent · US Expired

Derivatives of N-iminopyridinium betaines having anti-hypertensive and salidiuretic activity and their preparation

US4563467A · kind A · utility

13Cited by
1References
5Claims
0Family size

Assignee

Inventor

Key dates

Filing dateFeb 6, 1984
Grant dateJan 7, 1986
Priority date
Expiry dateFeb 6, 2004

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Derivatives of inner salts of aminopyridinium hydroxide and corresponding salts thereof comprising the general formuale I and II ##STR1## in which: R.sub.1 as selected from the group consisting of a hydrogen and a radical 2-furyl-methyl-amino; PA0 R.sub.2, R.sub.4 and R.sub.6 are all selected from the group consisting of a hydrogen atom, a C.sub.1 -C.sub.1 linear or branched lower alkyl radical and a phenyl radical; PA0 R.sub.3 is selected from the group consisting of a hydrogen or a carbamyl radical; PA0 R.sub.5 represents a hydrogen; and PA0 X.crclbar. represents a monobasic anion of a pharmaceutically acceptable acid.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.