Patent · US Expired

Substituted 5-hydroxy-2,3-dihydrobenzofurans and analogs thereof useful as anti-inflammatory agents

US4563476A · kind A · utility

4Cited by
0References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 21, 1983
Grant dateJan 7, 1986
Priority date
Expiry dateNov 21, 2003

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D409/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Substituted 5-hydroxy-2,3-dihydrobenzofuran and analogs such as the substituted 6-hydroxy-2,3-dihydrobenzopyrans were prepared from an appropriately substituted (5-hydroxy-2,3-dihydrobenzofuran-6-yl) formaldehyde or analog thereof with an aryl amine followed by reduction. These compounds were found to be potent topical anti-inflammatory agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.