Patent · US Expired

8-Oxo-2-oxa-1-azabicyclo(4.2.0)octane-3-carboxylic acids

US4574153A · kind A · utility

3Cited by
1References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 1, 1985
Grant dateMar 4, 1986
Priority date
Expiry dateMar 1, 2005

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D317/20
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Antibacterial activity is exhibited by compounds having the formula ##STR1## and pharmaceutically acceptable salts thereof, wherein, R.sub.1 is an acyl group derived from a carboxylic acid; PA0 R.sub.2 is hydrogen, methoxy, or formamido ##STR2## and one of R.sub.3 and R'.sub.3 is hydrogen and the other is ##STR3## and R.sub.4 is hydrogen alkyl, substituted alkyl, phenyl, substituted phenyl, phenylalkyl or (substituted phenyl)alkyl.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.