Patent · US Expired

Process for preparing 1-substituted-1,4-benzodiazepine derivatives

US4579685A · kind A · utility

0Cited by
1References
19Claims
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Assignee

Inventors

Key dates

Filing dateJul 27, 1984
Grant dateApr 1, 1986
Priority date
Expiry dateJul 27, 2004

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Improvement in the production of psychotropic 1-substituted-1,3-dihydro-1,4-benzodiazepin-2-ones starting from 2-(1-substituted)amino-benzophenonimines through novel intermediates of the formula: ##STR1## (wherein R is hydrogen, methyl or benzyl, R.sup.1 is C.sub.1 -C.sub.5 alkyl or phenyl-C.sub.1 -C.sub.5 alkyl, X and Y each is hydrogen or halogen and n is an integer of 1 to 2) with economical and industrial advantage.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.