Antihypertensive cyanoguanidines
US4579845A · kind A · utility
Assignee
Inventors
Key dates
| Filing date | Dec 8, 1983 |
| Grant date | Apr 1, 1986 |
| Priority date | — |
| Expiry date | Dec 8, 2003 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D405/06
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
This invention relates to novel tri-substituted guanidines linked to a piperidine ring. More specifically, it relates to cyanoguanidines of formula I ##STR1## wherein R.sub.1, R.sub.2, R.sub.3, R.sub.4 are substituents PA0 n is an integer of zero to 1 PA0 n' is an integer of zero to 1 PA0 A and B are --CH.sub.2 --, CHOH, --CO-- or a single bond as well as the acid addition salts thereof with a mineral or organic acid. The compounds have interesting pharmacological properties which make them useful as active ingredient of medicines, e.g. antihypertensives.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.