Patent · US Expired

Azole derivatives antimycotic agents which release the active compounds at a relatively high rate

US4585782A · kind A · utility

1Cited by

10References

10Claims

0Family size

Assignee

BAYER HEALTHCARE LLC · DE

Inventors

Manfred Plempel · Haan, DE
Manfred Bucheler · Overath, DE
Wolfgang Gau · Wuppertal, DE
Erik Regel
Karl H. Buchel · Burscheid, DE
Hans-Jurgen Ploschke · Wuppertal, DE

Key dates

Filing date	Feb 21, 1984
Grant date	Apr 29, 1986
Priority date	—
Expiry date	Feb 21, 2004

Classification

Technology area (CPC A)Human Necessities
CPC primaryA61K31/415
WIPO fieldPharmaceuticals
WIPO sectorChemistry

Abstract

The invention relates to antimycotic compositions comprising (1) an antimycotic effective amount of an azole derivative having antimycotic activity, said azole derivative being in the form of particles less than 4.mu. in size, (2) an acid and/or a buffer system consisting of an organic acid and a salt thereof to provide a pH of 3 to 4 or less in aqueous solution and (3) an inert pharmaceutical carrier. Also included in the invention are methods for the short term treatment of vaginal infections utilizing the compositions of the invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.