Patent · US Expired

Amidine benzodiazepines, methods for their use and intermediates

US4587244A · kind A · utility

1Cited by
0References
2Claims
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Assignee

Inventor

Key dates

Filing dateApr 10, 1985
Grant dateMay 6, 1986
Priority date
Expiry dateApr 10, 2005

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Fused tetracyclic benzodiazepines of the formula (I): ##STR1## where R.sup.1 is a cyclic amine such as 1-piperazine and R.sup.2 is H or a substituent as defined herein are useful as antiovulatory and contragestational agents. Also, methods for their synthesis, intermediates used in such synthesis, methods for use as medicaments and pharmaceutical compositions are described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.