Patent · US Expired

Derivatives of isoxazolo[4,5-c]quinoline(2H)-3-one and method of preparation and use as anxiolytic agents

US4588731A · kind A · utility

1Cited by
0References
21Claims
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Assignee

Inventors

Key dates

Filing dateJun 21, 1985
Grant dateMay 13, 1986
Priority date
Expiry dateJun 21, 2005

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D215/56
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Novel isoxazoloquinolinones of the formula ##STR1## wherein R is selected from the group consisting of hydrogen, fluorine, chlorine, bromine, alkyl and alkoxy of 1 to 5 carbon atoms, --NO.sub.2 and CF.sub.3 -- and R.sub.1 is phenyl optionally substituted by at least one member selected from the group consisting of halogen and alkyl and alkoxy of 1 to 5 carbon atoms having anxiolytic activity and their preparation and novel intermediates.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.