Patent · US Expired

Phospholipase A.sub.2 inhibition using 4,1-benzoxazepine-2-(3H)-ones

US4590187A · kind A · utility

1Cited by
6References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 19, 1984
Grant dateMay 20, 1986
Priority date
Expiry dateDec 19, 2004

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D267/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides certain novel 4,1-benzoxazepin-2(3H)-ones which are useful as inhibitors of phospholipase A.sub.2 and thus as inhibitors of arachidonate mobilization. These compounds are thus useful whenever it is medically necessary or desirable to inhibit the biosynthesis of the products of the arachidonic acid cascade.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.