Patent · US Expired

Preparation of penem derivatives and azetidinone intermediates

US4595539A · kind A · utility

3Cited by
9References
10Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJun 10, 1983
Grant dateJun 17, 1986
Priority date
Expiry dateJun 10, 2003

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D499/88
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Certain 2-substituted-2-penem-3-carboxylic acid compounds and pharmaceutically-acceptable salts thereof can be prepared from the appropriate xanthate or trithiocarbonate by desulfurization and addition of an electrophilic sulfur compound followed by halogenation and ring closure. The corresponding desulfurized and halogenated olefinic intermediates are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.