Patent · US Expired

Thiadiazole derivatives active on the central nervous system and pharmaceutical compositions

US4596802A · kind A · utility

5Cited by
2References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 11, 1985
Grant dateJun 24, 1986
Priority date
Expiry dateOct 11, 2005

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D285/135
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention relates to thiadiazole derivatives corresponding to the formula: ##STR1## in which R represents: a linear or branched alkyl group having from 1 to 5 carbon atoms; PA1 a cycloalkyl group having 5 or 6 carbon atoms; PA1 a phenyl group optionally substituted by 1 or 2 halogen atoms, preferably chlorine, by 1 or 2 lower alkyl or lower alkoxy groups, by 1 or 2 hydroxyl groups or by a nitro or trifluoromethyl group; PA1 a biphenylyl group; or PA1 an alpha-naphthyl group; and the pharmaceutically acceptable salts of the said derivatives. It also relates to a process for the preparation of the said derivatives and the pharmaceutical compositions in which they are present. The said derivatives act on the central nervous system.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.