Patent · US Expired

Process for preparing 2,2-bishalomethylpenam derivatives

US4599151A · kind A · utility

2Cited by
2References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 15, 1985
Grant dateJul 8, 1986
Priority date
Expiry dateMar 15, 2005

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention provides a process for preparing a 2,2-bishalomethylpenam derivative represented by the formula ##STR1## wherein R.sup.1 represents a lower alkyl group, aryl group, arylmethyl group, arylcarbonyl group or aryloxymethyl group, R.sup.2 represents a carboxyl-protecting group, X.sup.1 and X.sup.2 are the same or different and represent a halogen atom, the process being characterized in that a disulfide represented by the formula ##STR2## wherein R.sup.1, R.sup.2 and X.sup.1 are as defined above and R.sup.3 represents an aryl group or heterocyclic group is subjected to an electrolytic reaction in a solvent in the presence of a halogen acid and/or halogen salt.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.